Rakelin Injection 20ml

Long-acting non-sedating injectable calmative agent

COMPOSITION
Contains: Reserpine 0.5 mg/mL

ACTIONS
RAKELIN causes a rapid release of the nerve system transmitters norepinephrine and serotonin from bound stores in the brain, subjecting them to rapid destruction by the body's own enzyme, monoamine oxidase (MOA). While "bound" the stores are not available to MOA. Norepinephrine and serotonin have potent effects on the metabolism of the brain. High levels (especially of norepinephrine) cause stimulation of cerebral activity and anxiety. Lowered levels depress cerebral activity resulting in relaxation and calmness. Norepinephrine and serotonin, on release from the bound stores, undergo rapid destruction by MOA. The net depletion of these substances creates the calming and relaxing effects of RAKELIN. These effects continue for many days after administration, because levels are restored only slowly.

INDICATIONS
A calming agent to aid in the training and education of horses.
Rakelin should be used wherever a prolonged period of calm sedation is required. Rakelin is a useful aid in the handling of young horses and as a training aid where unfamiliar surroundings and unaccustomed stress may produce anxiety.

PRESENTATION
20 mL sterile glass multidose vial for intramuscular injection

STORAGE
Store below 25°C (Air Conditioning). Protect from light.

WARNINGS
RAKELIN may produce penile relaxation. Stallions which have been treated with RAKELIN should not be used to serve mares for at least 14 days following injection.
Meat Withholding Period: NOT TO BE USED in horses that will be slaughtered for human consumption.